Ownership
Private
Employees
~50
Therapeutic Areas
OncologyImmunologyNeurology
Stage
Phase 1
Preclinical
Phase 1
Phase 2
Phase 3
Approved
Modalities
Small molecules

858 Therapeutics General Information

858 Therapeutics has advanced its lead asset ETX‑19477—a potent and selective PARG inhibitor—into early-stage clinical trials for patients with advanced solid tumors. The company’s pipeline includes additional small molecule programs targeting novel nodes in cancer biology such as DNA repair mechanisms, innate immunity pathways, and RNA epigenetics. Recent financing rounds support ongoing clinical development.

Contact Information

Primary Industry
Biotech
Corporate Office
San Diego, California
United States

Drug Pipeline

ETX-19477
Phase 1
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Drug Asset 2
Phase X
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Drug Asset 3
Phase X
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Key Partnerships

OpenBench (collaboration on AI-driven small molecule drug discovery)

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858 Therapeutics Funding

Deal TypeDateAmountStatusStage
InvestmentSep 27, 2024$50.0MCompletedPhase 1
Early Stage VC (Series A)04-Jun-2020$38MCompletedPhase 1
Seed Round12-Feb-2019$8.5MCompletedStartup

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858 Therapeutics Financial Metrics