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1-[(2S)-4-(5-phenyl-1H-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine

Development stage: Unknown
Modality: Small Molecules

Overview

This compound is a synthetic small molecule belonging to the phenylpyridine class of organic compounds. It features a pyrazolo[3,4-b]pyridine core with a morpholine and methanamine substituent. The drug is experimental and has not been approved for any indication. Its primary known biological target is serine/threonine-protein kinase Chk1 (Checkpoint kinase 1), which plays a key role in cell cycle regulation and DNA damage response. Inhibition of Chk1 can sensitize tumor cells to DNA-damaging agents by abrogating cell cycle checkpoints, making this compound of interest as an anticancer agent in preclinical research settings[1].

Other names: 1-[(2S)-4-(5-phenyl-1H-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine

Targets

CHEK1 (Checkpoint kinase 1)

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