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N-[1-(aminomethyl)cyclopropyl]-3-(benzylsulfonyl)-N~2~-[(1S)-2,2,2-trifluoro-1-(4-hydroxyphenyl)ethyl]-L-alaninamide
- Development stage
- Unknown
- Modality
- Small Molecules
01
Overview
This compound is a synthetic small molecule belonging to the class of alpha amino acid amides. It is known as an experimental inhibitor of human cathepsin S—a lysosomal cysteine protease involved in antigen presentation and implicated in autoimmune diseases and cancer. The molecule acts as a covalent inhibitor by binding to the active site of cathepsin S. It has not been approved for any indication and has no reported clinical trials or marketed formulations[1][7][8].
- Other names
- N-[1-(aminomethyl)cyclopropyl]-3-(benzylsulfonyl)-N~2~-[(1S)-2,2,2-trifluoro-1-(4-hydroxyphenyl)ethyl]-L-alaninamide(2R)-N-[1-(aminomethyl)cyclopropyl]-3-phenylmethanesulfonyl-2-{[(1S)-2,2,2-trifluoro-1-(4-hydroxyphenyl)ethyl]amino}propanamide
02
Targets
CTSS (Cathepsin S)
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