Clinical trials
Full profile accessFollow clinical development from study design and recruitment through results.
- Trial phase
- Status
- Readouts
Drug intelligence / Profile preview
balanol analog 1
- Development stage
- Preclinical
- Modality
- Small Molecules
- Administration
- Not Specified (experimental; Likely In Vitro Or Ex Vivo Use)[4]
01
Overview
Balanol Analog 1 is a synthetic small molecule derivative of balanol, a fungal metabolite known for its potent inhibition of serine/threonine protein kinases. This analog has been specifically designed to enhance selectivity and potency against cyclic adenosine monophosphate-dependent protein kinase (PKA) over calcium- and phospholipid-dependent protein kinase (PKC). Structural studies show that it binds to the catalytic domain of PKA, stabilizing an intermediate conformation of the Gly-rich loop and disengaging key phosphoryl transfer residues. The compound acts as a competitive inhibitor at the ATP-binding site of these kinases. Its chemical formula is C20H22N2O5[2][3][4][5]. It remains an experimental drug candidate with no approved clinical indications.
- Other names
- Balanol Analog 1PD007822PD-007822PD 007822B1LB-1LB 1L
02
Targets
PKC (Protein kinase C family)PKA (Cyclic amp-dependent protein kinase)
Beyond the preview
Go deeper on balanol analog 1.
Explore the evidence, development activity, and competitive landscape with Gosset’s full data platform.
Indications & development
Full profile accessExplore development by indication, patient population, and geography.
- Indications
- Development status
- Countries
Licensing & deals
Full profile accessTrace asset ownership, licensing agreements, and commercial partnerships.
- Partners
- Deal terms
- Milestones
Patents & exclusivity
Full profile accessExplore the patent landscape and regulatory exclusivity around an asset.
- Patents
- Expiration dates
- Exclusivity
Competitive landscape
Full profile accessCompare development programs by target, modality, and indication.
- Competing assets
- Targets
- Development stage
Research & analysis
Full profile accessConnect source evidence and development news to your research questions.
- Publications
- News
- Analysis
Bring the full picture into focus.
See how Gosset can support your research on balanol analog 1.