Drug intelligence / Profile preview

bepotastine

Development stage
Approved
Lead developer
Mitsubishi Tanabe Pharma
Modality
Small Molecules
Administration
Ophthalmic, Oral
01

Overview

Bepotastine is a second-generation, non-sedating antihistamine used primarily in the treatment of allergic conjunctivitis and, in some countries, for allergic rhinitis and urticaria/pruritus. It acts as a selective antagonist of the histamine H1 receptor and also inhibits the release of histamine from mast cells. This dual action helps reduce symptoms such as ocular itching associated with allergies. Bepotastine is available in both ophthalmic (eye drop) and oral formulations. The drug was originally discovered by Ube Industries and co-developed with Tanabe Seiyaku; it is marketed under different brand names depending on region—Bepreve (ophthalmic solution) in the United States and Talion (oral/ophthalmic) in Japan. In the US, it was approved for ophthalmic use by the FDA in 2009[3][6][7].

Brand names
BepreveTalion
Other names
bepotastine besilate
02

Targets

HRH1 (Histamine H1 Receptor)

Beyond the preview

Go deeper on bepotastine.

Explore the evidence, development activity, and competitive landscape with Gosset’s full data platform.

Clinical trials

Full profile access

Follow clinical development from study design and recruitment through results.

  • Trial phase
  • Status
  • Readouts

Indications & development

Full profile access

Explore development by indication, patient population, and geography.

  • Indications
  • Development status
  • Countries

Licensing & deals

Full profile access

Trace asset ownership, licensing agreements, and commercial partnerships.

  • Partners
  • Deal terms
  • Milestones

Patents & exclusivity

Full profile access

Explore the patent landscape and regulatory exclusivity around an asset.

  • Patents
  • Expiration dates
  • Exclusivity

Competitive landscape

Full profile access

Compare development programs by target, modality, and indication.

  • Competing assets
  • Targets
  • Development stage

Research & analysis

Full profile access

Connect source evidence and development news to your research questions.

  • Publications
  • News
  • Analysis

Bring the full picture into focus.

See how Gosset can support your research on bepotastine.

Explore the full profile

Gosset Free

Get started with Gosset.

Enter your work email and we’ll be in touch with next steps.

Work email preferred.

Book a call