CRA_10656

CRA_10656 is a synthetic small molecule belonging to the phenylbenzimidazole class of organic compounds. Its chemical formula is C18H20N4O2, and it has been studied primarily as a selective inhibitor of trypsin-like serine proteases, particularly targeting the S1 site of these enzymes. Structural studies have demonstrated its binding to trypsin 1, indicating its potential utility in modulating protease activity for research or therapeutic purposes[1][4][9]. There is no evidence that it has advanced into clinical development for any specific disease.

Other names

2-{5-[amino(iminio)methyl]-1H-benzimidazol-2-yl}-6-isobutoxybenzenolate2-(2-hydroxy-3-isobutoxyphenyl)-1H-benzoimidazole-5-carboxamidine