Drug intelligence / Profile preview

diethylthiambutene

Development stage
Unknown
Modality
Small Molecules
Administration
Intramuscular, Subcutaneous, Intravenous
01

Overview

Diethylthiambutene is a synthetic opioid analgesic developed in the 1950s, primarily used as an anesthetic in veterinary medicine. It belongs to the thiambutene class of opioids and is structurally related to methadone. Its main use has been for anesthesia in animals, particularly in Japan. Diethylthiambutene acts as an agonist at opioid receptors, producing analgesia and sedation typical of opioids. Due to its high potential for abuse and lack of accepted medical use in humans, it is classified as a Schedule I controlled substance under both US law and international conventions[1][2][4].

Brand names
themalondiethibutin
Other names
thiambutenedietiltiambutenoN,N-diethyl-1-methyl-3,3-di-2-thienylallylamine
02

Targets

DOR (Opioid Receptor Delta 1)KOR (Kappa opioid receptor)MOR (Mu opioid receptor)

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