Drug intelligence / Profile preview

lipid-soluble vitamins for injection

Development stage
Unknown
Lead developer
Haisco Pharmaceutical Group
Modality
Small Molecules
Administration
Intravenous, Parenteral
01

Overview

**Lipid-soluble vitamins for injection** (also known as **Fat-Soluble Vitamins for Injection II**) is an approved intravenous nutritional supplement containing a combination of four essential fat-soluble vitamins: Vitamin A (retinol palmitate), Vitamin D2 (ergocalciferol), Vitamin E (tocopherol acetate), and Vitamin K1 (phytonadione). Developed by companies including Shanxi Pude Pharmaceutical and Haisco Pharmaceutical, this formulation is typically prepared as a lipid emulsion or lyophilized powder for reconstitution, designed to prevent and treat fat-soluble vitamin deficiencies in patients receiving parenteral nutrition. Once administered, the active components undergo metabolic activation to engage their respective biological pathways: Vitamin A metabolites bind to nuclear retinoic acid receptors (RARs) to regulate cell growth and differentiation; Vitamin D2 is converted to active calcitriol to bind the Vitamin D receptor (VDR) for calcium homeostasis; Vitamin E acts as a membrane-bound antioxidant; and Vitamin K1 serves as a cofactor for gamma-glutamyl carboxylase (GGCX) to activate blood coagulation factors. The product is widely approved and marketed in China for adult and pediatric patients requiring intravenous nutritional support.

Brand names
Lishi力时
Other names
Fat-Soluble Vitamins for Injection (II)Fat-Soluble Vitamins for Injection IIlipid-soluble vitamins for injection (II)注射用脂溶性维生素(II)注射用脂溶性维生素(Ⅱ)
02

Targets

F9 (Coagulation Factor IX)F7 (Coagulation Factor VII)F10 (Factor Xa)MGP (Matrix Gla protein)F2 (Thrombin)RARA (Retinoic acid receptor alpha)RARB (Retinoic acid receptor beta)RARG (Retinoic acid receptor gamma)VDR (Vitamin D receptor)VKORC1 (Vitamin K epoxide reductase complex subunit 1)GGCX (Vitamin K-dependent gamma-glutamyl carboxylase)

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