Drug intelligence / Profile preview

MRS8288

Development stage
Unknown
Lead developer
National Institutes of Health
01

Overview

MRS8288: sourced facts only. name: "Effects on ATPase activity of both ABCG2 and P-glycoprotein identified m-substituted N6-benzyl derivative 16 (MRS8288) as a dual inhibitor, with IC50 1.0 and 1.4 μM, respectively." [PMID:41703909]; target: "Effects on ATPase activity of both ABCG2 and P-glycoprotein identified m-substituted N6-benzyl derivative 16 (MRS8288) as a dual inhibitor, with IC50 1.0 and 1.4 μM, respectively." [PMID:41703909]; developer: "Laboratory of Cell Biology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892, United States." [PMID:41703909]

02

Targets

ABCG2 (Breast cancer resistance protein)

Beyond the preview

Go deeper on MRS8288.

Explore the evidence, development activity, and competitive landscape with Gosset’s full data platform.

Clinical trials

Follow clinical development from study design and recruitment through results.

  • Trial phase
  • Status
  • Readouts

Indications & development

Explore development by indication, patient population, and geography.

  • Indications
  • Development status
  • Countries

Licensing & deals

Trace asset ownership, licensing agreements, and commercial partnerships.

  • Partners
  • Deal terms
  • Milestones

Patents & exclusivity

Explore the patent landscape and regulatory exclusivity around an asset.

  • Patents
  • Expiration dates
  • Exclusivity

Competitive landscape

Compare development programs by target, modality, and indication.

  • Competing assets
  • Targets
  • Development stage

Research & analysis

Connect source evidence and development news to your research questions.

  • Publications
  • News
  • Analysis

Bring the full picture into focus.

See how Gosset can support your research on MRS8288.

Gosset Free

Get started with Gosset.

Enter your corporate email.

Work email preferred.

Book a call