Drug pipeline
Full profile accessExplore the programs pursuing this target and their development progress.
- Drug candidates
- Developers
- Development stage
Target intelligence / Profile preview
Deshydroxyethoxy Ticagrelor (AR-C124910XX)
- Target
- AR-C124910XX
- Molecular classification
- Nucleoside analogue, Receptor antagonist, P2Y12 receptor antagonist
01
Overview
AR-C124910XX is the principal active metabolite of ticagrelor, a widely used antiplatelet medication. It is formed in vivo by O-deethylation of ticagrelor and retains pharmacological activity similar to its parent compound. AR-C124910XX acts as an inhibitor of the P2Y12 receptor on platelets, preventing ADP-induced platelet aggregation and reducing thrombotic risk in patients with acute coronary syndromes or other cardiovascular conditions treated with ticagrelor.
- Other names
- AR-C124910XXTicagrelor active metaboliteTicargrelor Impurity D/G-d7Fluometacyl
02
Mechanism of action
Reversible P2Y12 receptor antagonist
03
Biological functions
Inhibition of platelet aggregationP2Y12 receptor inhibition
04
Disease associations
Cardiovascular diseaseAcute coronary syndromesThrombotic risk
05
Interacting drugs
Ticagrelor
Beyond the preview
Go deeper on Deshydroxyethoxy Ticagrelor (AR-C124910XX).
Explore the evidence, development activity, and competitive landscape with Gosset’s full data platform.
Clinical trials
Full profile accessFollow the clinical studies evaluating therapies directed at this target.
- Trial design
- Status
- Readouts
Competitive landscape
Full profile accessCompare approaches across drug candidates, modalities, and indications.
- Programs
- Modalities
- Indications
Literature & evidence
Full profile accessInvestigate the research and source evidence behind target biology and development.
- Publications
- Sources
- Analysis
Patents
Full profile accessExplore patent activity around therapies and technologies addressing this target.
- Patents
- Assignees
- Technologies
Research & analysis
Full profile accessConnect target biology, drug development, and emerging evidence in your research.
- Biology
- Development news
- Analysis
Bring the full picture into focus.
See how Gosset can support your research on Deshydroxyethoxy Ticagrelor (AR-C124910XX).